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CAS No.: 841290-80-0
Synonyms: R406;R406 Free Base;Tamatinib
R406 is an inhibitor of Syk with IC50 of 41 nM.
生物活性
靶点 | Syk IC50:41nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01725230 | Rheumatoid Arthritis | Phase 1 | Completed | - | United States, Kansas ... more >> Research Site Overland Park, Kansas, United States Collapse << |
NCT01208155 | Bioavailability ... more >> Pharmacokinetics Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> Research Site Overland Park, Kansas, United States Collapse << |
NCT01245790 | Rheumatoid Arthritis ... more >> Renal Impairment Collapse << | Phase 1 | Completed | - | United States, Florida ... more >> Research Site Orlando, Florida, United States Collapse << |
实验方案
技术信息
CAS号 | 841290-80-0 | 储存条件 |
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分子式 | C22H23FN6O5 | 运输 | 蓝冰 | |||||||||||
分子量 | 470.45 | 别名 | R406;R406 Free Base;Tamatinib | |||||||||||
溶解度 |
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动物实验配方 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01725230 | Rheumatoid Arthritis | Phase 1 | Completed | - | United States, Kansas ... more >> Research Site Overland Park, Kansas, United States Collapse << |
NCT01208155 | Bioavailability ... more >> Pharmacokinetics Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> Research Site Overland Park, Kansas, United States Collapse << |
NCT01245790 | Rheumatoid Arthritis ... more >> Renal Impairment Collapse << | Phase 1 | Completed | - | United States, Florida ... more >> Research Site Orlando, Florida, United States Collapse << |
NCT01355354 | Healthy Volunteers ... more >> Rheumatoid Arthritis Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT01197781 | Drug Drug Interactions ... more >> Healthy Volunteers Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> Recruiting Site Overland Park, Kansas, United States Collapse << |
NCT01387308 | Healthy | Phase 1 | Completed | - | United States, Kansas ... more >> Research Site Overland Park, Kansas, United States Collapse << |
NCT01276262 | Scientific Terminology Rheumat... more >>oid Arthritis, Healthy Female Volunteers, Pharmacokinetics, Oral Contraceptive, Drug-drug Interaction Laymen Terminology Level of Oral Contraceptive in Blood, Oral Contraceptive, Rheumatoid Arthritis, Drug -Drug Interaction Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT01336218 | Rheumatoid Arthritis ... more >> Healthy Volunteers Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> Research Site Overland Park, Kansas, United States Collapse << |
NCT01598571 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Ruddington, Nottingham, United Kingdom Collapse << |
NCT01311622 | Rheumatoid Arthritis ... more >> Healthy Subjects Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT01682408 | Pharmacokinetics | Phase 1 | Completed | - | United States, Kansas ... more >> Overland Park, Kansas, United States Collapse << |
NCT01222455 | Hepatic Impairment ... more >> Healthy Volunteers Pharmacokinetics Amount of R406 in Blood Collapse << | Phase 1 | Completed | - | United States, Florida ... more >> Research Site Orlando, Florida, United States Collapse << |
NCT01645085 | Healthy Volunteers | Phase 1 | Completed | - | United States, Kansas ... more >> Overland Park, Kansas, United States Collapse << |
靶点 | Description | IC50 |
---|---|---|
Syk | IC50:41nM |
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